Wednesday, August 17, 2011

Enantioselective α-Arylation of Carbonyls via Cu(I)-Bisoxazoline Catalysis

The enantioselective α-arylation of both lactones and acyl oxazolidones has been accomplished using a combination of diaryliodonium salts and copper catalysis. These mild catalytic conditions provide a new strategy for the enantioselective construction and retention of enolizable α-carbonyl benzylic stereocenters, a valuable synthon for the production of medicinal agents.


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